Paʻu 7P paʻu (1890208-58-8) vitio
Paʻu 7P faʻamalosi (1890208-58-8) faʻamatalaga
Faʻasologa o le 7P paʻu o loʻo faʻaleleia ai le fua o le matua mai i meaola faʻatoʻaga e maua mai i le hippocampus, corbex cerebral, ma le retina. I se faʻataʻitaʻiga manu o le manua o le nerve opic, o le elemene Raw 7P o loʻo faʻaalia ai le faatupuina o le vaʻa-43 axons lelei, e faʻamaonia ai o le in vitro o le gaioiga fou o le Raw Compound 7P powder e faaliliuina i le stimulation o le axon regeneration in vivo.further optimization of Faʻaaogaina o le eletise 7P ma le maualuga o faʻamautuga e faʻaaogaina ai le toe faʻafouina o le axon i totonu o vivo, o le a maua ai se faavae faʻavae mo taumafaiga i le lumanaʻi e faʻaleleia ai togafitiga togafitiga.
mata 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Vaega 7P) paʻu (1890208-58-8) Sfaʻamatalaga
Igoa oloa | 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Paʻu 7P paʻu) |
Suafa Suafa | 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Raw Compound 7P paʻu) |
faʻailogaina Nma | Laʻu Faʻamalosi 7P paʻu |
Vailaʻau Vailaʻau | Nootropic Drugs |
Numera CAS | 1890208-58-8 |
InChIKey | NAXWKPFXCOBXLE-UHFFFAOYSA-N |
Molecular Famulamu | C22H23N3O5S |
Molecular Wvalu | 441.508g |
Masima Monoisotopic | 440g / mol |
Mea faʻamafanafana | N / A |
Ftoe ola Pmanogi | N / A |
Half-Life Biological | N / A |
lanu | Paʻu paʻu |
Sfaʻamalosia | sina solu i totonu o le vai ma le ethanol. |
Storage Tsuauu | Teu i le vevela o le potu, i totonu o fagu faʻamaufaʻailoga, aloese mai le vevela malosi ma le malamalama |
Afaʻasologa | • Faateleina le faʻatulagaga • Faaleleia lagona • Fesoasoani i le tauva vaivai • Puipuia le faʻamaʻiina i totonu o le faiʻai • Taulimaina le faaleagaina o le faia o le ava |
mata Faʻatasi 7P paʻu (1890208-58-8) Faamatalaga
Raw Compound 7P (2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide) paʻu lea e faʻalauiloa ai le olaola o le neurite tuputupu aʻe muamua neurons na mafua mai i le hippocampus , cerebral cortex, ma le retina. I totonu o se manu faʻataʻitaʻi o manuʻa neura o le neura, Raw Compound 7P paula na faʻaalia e faʻatupu ai le tuputupu ae o va-43 lelei axon, e faʻailoa mai ai o le in vitro neurite outgrowth activity o Raw Compound 7P paʻu faʻaliliuina i le faʻaosofia o le toe faʻafouina axon i vivo.further optimization o Raw Compound 7P efuefu ma elucidation o auala ia e faʻaosofia ai le toe faʻafouina o le axon i le vivo o le a maua ai se faʻavae talafeagai mo lumanaʻi taumafaiga e faʻaleleia togafitiga togafitiga.
Faaaogaina o le 7P Faʻatasi paʻu (1890208-58-8)
O le 7p (2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide) na faaalia ai le maualuga o le gaioiga e faasaga i potu o le kanesa. I se faʻataʻitaʻiga o le gutu o le xenograft faʻapipiʻiina i le cellules o le HeLa, o le 7p na faʻaalia le puipuia o le toto o le tino. O le suʻesuʻeina o talafaasolopito o masini vailaau oona na faaalia ai o 7p na faʻaleleia le microstructure i se faʻatonuga-faalagolago. O le 7p faʻatele na faʻapupulaina foi le tele o lela o le HeLa i le G0 / G1 ma le S ma faʻaititia ai le tele o le G2 / M-phase. O aʻafiaga o le 7p i luga o le C-caspase-3, C-caspase-9, Bcl-2 ma le faʻamatalaga Paʻu i le cellules o le HeLa na fuafuaina foi.
O le suʻega o le polymerization o le Tulinulin, suʻesuʻega o le immunofluorescence, faʻataʻitaʻiga faataamilosaga o le tino ma le faʻatauvaga o le tui tui-tui faʻamaonia na faʻamaonia ai o 7p o se inhibitor site o le pulchicine o le tubulin.
faamanuiaga of Faʻatasi 7P paʻu (1890208-58-8)
Faʻatasi le 7p faʻateleina le faʻafouina o le masini vili
Toe faaleleia le nerve faaleagaina
fautuaina Faʻatasi 7P paʻu (1890208-58-8) Faʻailoga
O le 7p faʻamaonia le 100% faʻasaina o le parasitemia i le aso 4 i le tele o doses (100, 50, ma 25 mg / kg) na tuʻuina mo aso e fa aso, ae i 100 mg / kg, na ola uma mice ma na faʻamalolo, ao 50 mg / kilokalama, tolu o le 5 muni na ola ma lua moa sa malolo, ma i le 25 mg / kg, e leai se muse na sao